ペチジン
出典: フリー百科事典『ウィキペディア（Wikipedia）』 (2023/05/06 09:00 UTC 版)
関連項目
歴史
初の合成鎮痛薬として、1939年にドイツで開発された。日本で薬価収載されたのは原末（経口薬）が1955年1月[9]、注射液が1956年9月である[10]。
関連項目
参考文献
- 伊藤勝昭ほか編集 『新獣医薬理学 第二版』 近代出版 2004年 ISBN 4874021018
- ^ “Demerol, Pethidine (meperidine) dosing, indications, interactions, adverse effects, and more”. Medscape Reference. WebMD. 2014年4月9日閲覧。
- ^ Shipton, E (March 2006). “Should New Zealand continue signing up to the Pethidine Protocol?” (PDF). The New Zealand Medical Journal 119 (1230): U1875. PMID 16532042. オリジナルの2014年4月8日時点におけるアーカイブ。.
- ^ a b c d Latta, KS; Ginsberg, B; Barkin, RL (January–February 2002). “Meperidine: a critical review.”. American Journal of Therapeutics 9 (1): 53–68. doi:10.1097/00045391-200201000-00010. PMID 11782820.
- ^ a b MacPherson, RD; Duguid, MD (2008). “Strategy to Eliminate Pethidine Use in Hospitals” (PDF). Journal of Pharmacy Practice and Research 38 (2): 88–89.
- ^ Mather, LE; Meffin, PJ (September–October 1978). “Clinical pharmacokinetics of pethidine.”. Clinical Pharmacokinetics 3 (5): 352–68. doi:10.2165/00003088-197803050-00002. PMID 359212.
- ^ a b Rossi, S, ed (2013). Australian Medicines Handbook (2013 ed.). Adelaide: The Australian Medicines Handbook Unit Trust. ISBN 978-0-9805790-9-3
- ^ Michaelis, Martin; Schölkens, Bernward; Rudolphi, Karl (April 2007). “An anthology from Naunyn-Schmiedeberg's archives of pharmacology”. Naunyn-Schmiedeberg's Archives of Pharmacology (Springer Berlin) 375 (2): 81–84. doi:10.1007/s00210-007-0136-z. PMID 17310263.
- ^ Kaiko, Robert F.; Kathleen M. Foley; Patricia Y. Grabinski; George Heidrich; Ada G. Rogers; Charles E. Inturrisi; Marcus M. Reidenberg (February 1983). “Central Nervous System Excitatory Effects of Meperidine in Cancer Patients”. Annals of Neurology (Wiley Interscience) 13 (2): 180–185. doi:10.1002/ana.410130213. PMID 6187275.
- ^ a b c d e “オピスタン原末 添付文書” (2015年4月). 2016年4月5日閲覧。
- ^ a b c d e “ペチジン塩酸塩注射液35mg／ペチジン塩酸塩注射液50mg 添付文書” (2015年7月). 2016年11月6日閲覧。
- ^ http://www.deadiversion.usdoj.gov/fed_regs/quotas/2014/fr0825.htm
- ^ “Parenteral opioids for labor pain relief: A systematic review - American Journal of Obstetrics & Gynecology”. www.ajog.org. 2015年7月11日閲覧。
- ^ “Narcotics for Pain During Labor: Types & Side Effects”. 2015年6月20日閲覧。
- ^ “WHO en:Template:! Parenteral opioids for maternal pain relief in labour”. apps.who.int. 2015年6月20日閲覧。
- ^ “Pain relief in labour - Pregnancy and baby guide - NHS Choices”. www.nhs.uk. 2015年6月20日閲覧。
- ^ Blueprints - Family Medicine (3rd edition)
- ^ Baselt, R. (2008). Disposition of Toxic Drugs and Chemicals in Man (8 ed.). Foster City, CA: Biomedical Publications. pp. 911-914.
- ^ Package insert for meperidine hydrochloride, Boehringer Ingelheim, Ridgefield, CT, 2005.
- ^ Brody, Jane (2007年2月27日). “A Mix of Medicines That Can Be Lethal”. New York Times 2009年2月13日閲覧. "The death of Libby Zion, an 18-year-old college student, in a New York hospital on March 5, 1984, led to a highly publicized court battle and created a cause célèbre over the lack of supervision of inexperienced and overworked young doctors. But only much later did experts zero in on the preventable disorder that apparently led to Ms. Zion’s death: a form of drug poisoning called serotonin syndrome."
- ^ Bronwen Bryant and Kathleen Knights (2010). Pharmacology for Health Professionals, 3rd Edition. Chatswood: Mosby Australia. ISBN 978-0-7295-3929-6
- ^ Koczmara, C; Perri, D; Hyland, S; Rousseaux, L (2005). “Meperidine (Demerol) safety issues”. Official Journal of the Canadian Association of Critical Care Nurses 16 (1): 8–12. ISSN 1201-2580 2014年1月11日閲覧。.
- ^ Laurence, Brunton (2010). Goodman & Gilman's pharmacological basis of therapeutics (12th ed.). McGraw-Hill. p. 549. ISBN 0071624422
- ^ http://www.fass.se/LIF/produktfakta/artikel_produkt.jsp?NplID=19741206000040&DocTypeID=3&UserTypeID=0
- ^ Wagner, Larry E., II; Michael Eaton; Salas S. Sabnis; Kevin J. Gingrich (November 1999). “Meperidine and Lidocaine Block of Recombinant Voltage-Dependent Na+ Channels: Evidence that Meperidine is a Local Anesthetic”. Anesthesiology (Lippincott Williams & Wilkins) 91 (5): 1481–1490. doi:10.1097/00000542-199911000-00042. PMID 10551601.
- ^ a b c Izenwasser, Sari; Amy Hauck Newman; Brian M. Cox; Jonathan L. Katz (January–February 1996). “The cocaine-like behavioral effects of meperidine are mediated by activity at the dopamine transporter”. European Journal of Pharmacology (Elsevier) 297 (1–2): 9–17. doi:10.1016/0014-2999(95)00696-6. PMID 8851160.
- ^ Lomenzo, Stacey A.; Jill B. Rhoden; Sari Izzenwasser; Dean Wade; Theresa Kopajtic; Jonathan L. Katz; Mark L. Trudell (2005-03-05). “Synthesis and Biological Evaluation of Meperdine Analogs at Monoamine Transporters”. Journal of Medicinal Chemistry (American Chemical Society) 48 (5): 1336–1343. doi:10.1021/jm0401614. PMID 15743177.
- ^ a b c d “Demerol: Is It the Best Analgesic?” (PDF), Pennsylvania Patient Safety Reporting Service Patient Safety Advisory (Pennsylvania Patient Safety Authority) 3 (2), (June 2006) 2013年4月15日閲覧。
- ^ Davis, Sharon (2004年8月). “Use of pethidine for pain management in the emergency department: a position statement of the NSW Therapeutic Advisory Group”. New South Wales Therapeutic Advisory Group. 2007年1月17日閲覧。
- ^ a b c Latta, Kenneth S.; Brian Ginsberg; Robert L. Barkin (January–February 2002). “Meperidine: A Critical Review”. American Journal of Therapeutics (Lippincott Williams & Wilkins) 9 (1): 53–68. doi:10.1097/00045391-200201000-00010. PMID 11782820.
- ^ “In Brief”. NPS Radar. National Prescribing Service (2005年12月). 2009年12月22日閲覧。
- ^ Walker, Diana J.; James P. Zacny (June 1999). “Subjective, Psychomotor, and Physiological Effects of Cumulative Doses of Opioid µ Agonists in Healthy Volunteers”. The Journal of Pharmacology and Experimental Therapeutics (American Society for Pharmacology and Experimental Therapeutics) 289 (3): 1454–1464. PMID 10336539.
- ^ Molloy, A (2002). “Does pethidine still have a place in therapy?” (PDF). Australian Prescriber (NPS MedicineWise) 25 (1): 12–13.
- ^ Gilson AM, Ryan KM, Joranson DE, Dahl JL (2004). “A reassessment of trends in the medical use and abuse of opioid analgesics and implications for diversion control: 1997-2002”. J Pain Symptom Manage 28 (2): 176–188. doi:10.1016/j.jpainsymman.2004.01.003. PMID 15276196.
- ^ Joranson DE, Gilson AM (2005). “Drug crime is a source of abused pain medications in the United States”. J Pain Symptom Manage 30 (4): 299–301. doi:10.1016/j.jpainsymman.2005.09.001. PMID 16256890.
- ^ a b Lexicon of alcohol and drug terms. Geneva: World Health Organization. (1994). ISBN 92-4-154468-6
- ^ http://pubs.acs.org/doi/suppl/10.1021/jm0401614/suppl_file/jm0401614_s.pdf
- ^ Lomenzo, S.; Rhoden, J.; Izenwasser, S.; Wade, D.; Kopajtic, T.; Katz, J.; Trudell, M. (2005). “Synthesis and biological evaluation of meperidine analogues at monoamine transporters”. Journal of Medicinal Chemistry 48 (5): 1336–1343. doi:10.1021/jm0401614. PMID 15743177.
- ^ Lomenzo, S.; Izenwasser, S.; Gerdes, R. M.; Katz, J. L.; Kopajtic, T.; Trudell, M. L. (1999). “Synthesis, dopamine and serotonin transporter binding affinities of novel analogues of meperidine”. Bioorganic & Medicinal Chemistry Letters 9 (23): 3273–3276. doi:10.1016/S0960-894X(99)00606-X.
- ^ Rhoden, J. B.; Bouvet, M.; Izenwasser, S.; Wade, D.; Lomenzo, S. A.; Trudell, M. L. (2005). “Structure-activity studies of 3'-4'-dichloro-meperidine analogues at dopamine and serotonin transporters”. Bioorganic & Medicinal Chemistry 13 (19): 5623–5634. doi:10.1016/j.bmc.2005.05.025. PMID 15993612.
- ^ Gu, X.; Izenwasser, S.; Wade, D.; Housman, A.; Gulasey, G.; Rhoden, J. B.; Savoie, C. D.; Mobley, D. L. et al. (2010). “Synthesis and structure–activity studies of benzyl ester meperidine and normeperidine derivatives as selective serotonin transporter ligands”. Bioorganic & Medicinal Chemistry 18 (23): 8356. doi:10.1016/j.bmc.2010.09.060.
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